平安! 发表于 2011-11-9 19:57
* `% h$ `. _, o7 DPazopanib (100 mg/kg/day free base equivalent) 4 l( r7 _( Q" J: I1 B6 ]8 F/ S
这是个已经在美国上市的老药了,能下载到正式药物使用说明书英文版。2 c& U: ~% Z$ w2 s! |1 r
搜索了一下,原料一大堆。% D% u) i3 d& y. M8 i2 D* ?5 B% r
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对不起!100mg/kg是用于移植瘤的,我弄错了。: r/ C9 D3 j3 _$ f; h
& K4 E( h7 w) h1 W' V4 k" D以下是正版说明书的推荐用量。! G) {; Y) Q- a" a! V, z& y- _2 n9 j
* ?) K1 y' e, J* _2 A--------------------- DOSAGE AND ADMINISTRATION ----------------
5 l) v$ N" C+ u1 [% w1 B7 k, W1 r* 800 mg orally once daily without food (at least 1 hour before or 2 hours after a meal). (2.1) " |) N: K# A0 v" _) }
* Baseline moderate hepatic impairment – 200 mg orally once daily. Not recommended in patients with severe hepatic impairment. (2.2) 6 ]( h% j- n3 R# S* ?, L6 `
---------------------DOSAGE FORMS AND STRENGTHS --------------
, c7 N' h- I9 u! M9 G# n/ j" I200 mg tablets. (3)
: h; b6 q) t5 z-------------------------------CONTRAINDICATIONS------------------------ |