平安! 发表于 2011-11-9 19:57
! | G8 ]& o6 q6 rPazopanib (100 mg/kg/day free base equivalent) 8 y1 }, a' ~ K9 _3 h) s( m% ~: c
这是个已经在美国上市的老药了,能下载到正式药物使用说明书英文版。* [3 |8 ]/ v/ W$ [0 {% @, @
搜索了一下,原料一大堆。
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/ [+ W$ Z; R% t. }* B对不起!100mg/kg是用于移植瘤的,我弄错了。! Q9 D0 _1 i/ Z5 W m
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以下是正版说明书的推荐用量。
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& Q8 ? [" P- `' ?, k. A--------------------- DOSAGE AND ADMINISTRATION ----------------" h$ v* |' U V+ D' ^" p$ R
* 800 mg orally once daily without food (at least 1 hour before or 2 hours after a meal). (2.1)
. }% b9 t) ]1 l8 Z7 A* Baseline moderate hepatic impairment – 200 mg orally once daily. Not recommended in patients with severe hepatic impairment. (2.2) ' J' J7 Y; L$ p2 I& I! p- d+ q! ^
---------------------DOSAGE FORMS AND STRENGTHS --------------% G( ]8 v% B K I
200 mg tablets. (3)
7 K; ^% R2 ?' B2 J5 Z-------------------------------CONTRAINDICATIONS------------------------ |