平安! 发表于 2011-11-9 19:57 , X0 f' Q- \$ }5 x
Pazopanib (100 mg/kg/day free base equivalent)
9 t- C6 C$ a | _ 这是个已经在美国上市的老药了,能下载到正式药物使用说明书英文版。3 `8 Q" s) M8 s8 R/ {" o U' i
搜索了一下,原料一大堆。9 h# A+ ], L. j" o9 n6 C! l
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对不起!100mg/kg是用于移植瘤的,我弄错了。8 E/ E; V' b- @0 h/ p$ Z
! ~5 X# h) n: U# d2 T以下是正版说明书的推荐用量。7 ]" z! a$ d1 G7 [$ U$ n2 F5 o( ]0 V
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--------------------- DOSAGE AND ADMINISTRATION ----------------3 I3 M Q+ J& [# d+ `$ a
* 800 mg orally once daily without food (at least 1 hour before or 2 hours after a meal). (2.1)
3 [# G* u+ Y H" Z* Baseline moderate hepatic impairment – 200 mg orally once daily. Not recommended in patients with severe hepatic impairment. (2.2) - D8 U) u) r4 T" a* c& `
---------------------DOSAGE FORMS AND STRENGTHS --------------* @6 L1 S Y p0 R
200 mg tablets. (3) ' N7 D. D' _4 c9 l6 U8 u
-------------------------------CONTRAINDICATIONS------------------------ |