平安! 发表于 2011-11-9 19:57
4 w+ K' ]) S% N2 JPazopanib (100 mg/kg/day free base equivalent) : Z+ o8 n( ~' R( ? j
这是个已经在美国上市的老药了,能下载到正式药物使用说明书英文版。* A8 a; F( c0 u0 I, U
搜索了一下,原料一大堆。! J; R7 \; d2 S" W
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对不起!100mg/kg是用于移植瘤的,我弄错了。4 C. Z/ n/ ]1 E9 o$ T3 o+ L
+ q+ ]0 e8 q3 H% j& B以下是正版说明书的推荐用量。
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1 p+ a) T0 _: {5 E--------------------- DOSAGE AND ADMINISTRATION ----------------
9 v: V2 B$ Q/ X+ U- c* 800 mg orally once daily without food (at least 1 hour before or 2 hours after a meal). (2.1)
% {) ?6 H5 r$ Z+ x* g* Baseline moderate hepatic impairment – 200 mg orally once daily. Not recommended in patients with severe hepatic impairment. (2.2)
+ d/ E9 @ G2 T---------------------DOSAGE FORMS AND STRENGTHS --------------
" q0 p% \& e Z' y4 `" X. ^: f( O/ k200 mg tablets. (3)
6 M+ B8 ?+ H5 ?4 C* V7 K-------------------------------CONTRAINDICATIONS------------------------ |